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Cisapride

(CAS: 81098-60-4)

Suppliers of Cisapride

Company Name Email Tel Country
Abcam [email protected] (888) 77-ABCAM (22226) USA

Fax: (877) 774-8286 / (617) 577-4201Purity: Brand:

Price and Availability: USD69/10mg ()

CHEMSCENE, LLC [email protected] 732-484-9848 USA

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Clearsynth Labs Limited [email protected] Worldwide Helpline No. +1-415-685-4395; US & Canada (Toll-free) : +1-800-650-8239; Europe : +44-20-3286-0885; India : +91-22-26355700 India

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Price and Availability: USD200/25mg ()

MedChemexpress Co., Ltd. [email protected] 609-228-6898 USA

Fax: 609-228-5909Purity: >98% Brand:

Price and Availability: USD60/10mg (In stock) USD95/50mg (In stock) USD150/100mg (In stock) USD240/200mg (In stock)
Quality Control & MSDS Files: LCMS HNMR MSDS

Santa Cruz Biotechnology, Inc. [email protected] Toll Free: 800-457-3801 Phone: 214-902-3900 USA

Fax: 214-358-6070Purity: Brand:

Price and Availability: USD115/10mg ()

Shanghai Everchem Co., Ltd. [email protected],[email protected] +86 (29) 8132-5371 China

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Shanghai Haoyuan Chemexpress Co., Ltd. [email protected] +86 (21) 5187-0955 / +86 (21) 5895-5995 China

Fax: +86 (21) 5895-5996Purity: >98% Brand:

Price and Availability: USD75/10mg (Get quote) USD300/50mg (Get quote)

Target Molecule Corp. [email protected] (857) 239-0968 USA

Fax: 857-239-8801Purity: .98 Brand: TargetMol

Price and Availability: USD20/2mg () USD78/10mg () USD156/25mg ()

Tocris Bioscience Inc. [email protected] +1 (636) 207-7651 USA

Fax: +1 (636) 207-7683Purity: Brand:

Price and Availability: USD119/10mg ()

Toronto Research Chemicals Inc. [email protected] +1 (416) 665-9696 Canada

Fax: +1 (416) 665-4439Purity: Brand:

Price and Availability: USD115/10mg ()

Zhejiang Ouhua Chemical Imp. & Exp. Co., Ltd. [email protected] +86 (576) 8882-6717 China

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Background Information of Cisapride

Cisapride(R 51619) is a nonselective 5-HT4 receptor agonist, it is also a potent human ether-à-go-go-related gene (hERG) potassium channel inhibitor. IC50 Value: 0.14 μM(EC50 for 5-HT4 receptor) [1]; 9.8 μM (Kv4.3) [2] Target: 5-HT4 Receptor in vitro: Cisapride showed higher inhibitory effects on a hERG current, as indicated by its IC50 of 9.4 × 10-9 M [1].

Solubility of Cisapride

Solubility Sources
DMSO MedChemexpress Co., Ltd.

Storage Condition of Cisapride

Storage Condition Sources

MSDS Information

MSDS Sources
MedChemexpress Co., Ltd.

Quality Control and Spectral Data

QC Reports Sources
[LCMS] [HNMR] MedChemexpress Co., Ltd.

Mechanism and Indications

Signaling Pathways Neuronal Signaling GPCR/G Protein
Target 5-HT Receptor
Research Area Neurological Disease
Indications Hypoglycemia Constipation

Clinical Information

Product Name Sponsor & Collaborators Indications Start Date End Date Phase
Cisapride The Procter & Gamble Co Hypoglycemia 2008/2/29 2008/7/31 Phase 2 Clinical
Cisapride Procter & Gamble Pharmaceuticals Inc Constipation 2007/7/31 2008/7/31 Phase 2 Clinical
Cisapride Mayo Foundation 2005/1/31 2005/12/31 Phase 2 Clinical
Cisapride - Launched

Chemical Information

M.Wt Formula CAS No. Synonyms
465.95 C23H29ClFN3O4 81098-60-4 R 51619;(±)-Cisapride; 4-amino-5-chloro-N-((3S,4R)-1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide

Structure Information of Cisapride

Smiles ClC1=C(N)C=C(OC)C(C(N[[email protected]]2[[email protected]@H](OC)CN(CCCOC3=CC=C(F)C=C3)CC2)=O)=C1
InChI InChI=1S/C23H29ClFN3O4/c1-30-21-13-19(26)18(24)12-17(21)23(29)27-20-8-10-28(14-22(20)31-2)9-3-11-32-16-6-4-15(25)5-7-16/h4-7,12-13,20,22H,3,8-11,14,26H2,1-2H3,(H,27,29)/t20-,22+/m1/s1

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Chemical and Physical Properties

Appearance:White to off-white Solid Melting point:
Boiling point: Flash Point:
Water Solubility: Solubility:
Density: Merck:
BRN: Refractive Index:
Vapour: EINECS:279-689-7
Optical Rotation: alpha:

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