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VT-464 (racemate)

(CAS: 1375603-36-3)

Suppliers of VT-464 (racemate)

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Apexbio Technology LLC [email protected] +1-832-696-8203 USA

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Price and Availability: USD332/5mg () USD475/10mg () USD1425/50mg () USD1995/100mg ()

Ark Pharm, Inc. [email protected] +1 (847) 367-3680 USA

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BOC Sciences [email protected] 1-631-504-6093

Fax: 1-631-614-7828Purity: 98% Brand: BOC Sciences

CHEMSCENE, LLC [email protected] 732-484-9848 USA

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Price and Availability: USD420/5mg () USD600/10mg ()

MedChemexpress Co., Ltd. [email protected] 609-228-6898 USA

Fax: 609-228-5909Purity: Brand:

Price and Availability: USD420/5mg () USD600/10mg ()
Quality Control & MSDS Files: MSDS CoA LCMS

Shanghai Haoyuan Chemexpress Co., Ltd. [email protected] +86 (21) 5187-0955 / +86 (21) 5895-5995 China

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Price and Availability: USD420/5mg () USD600/10mg ()

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Background Information of VT-464 (racemate)

VT-464 racemate is the racemate form of VT-464, which is a potent CYP17 lyase inhibitor(h-Lyase IC50=69 nM)inhibition. IC50 value: 69 nM(VT-464, h-CYP17 Lyase) [1] Target: CYP17 Lyase inhibitor in vitro: VT-464, a non-steroidal small molecule inhibits androgen production without mineralocorticoid excess or cortisol depletion by selective inhibition of CYP17 17,20-lyase.

Solubility of VT-464 (racemate)

Solubility Sources
DMSO MedChemexpress Co., Ltd.

Storage Condition of VT-464 (racemate)

Storage Condition Sources

MSDS Information

MSDS Sources
MedChemexpress Co., Ltd.

Quality Control and Spectral Data

QC Reports Sources
[CoA] [LCMS] MedChemexpress Co., Ltd.

Mechanism and Indications

Signaling Pathways Metabolic Enzyme/Protease
Target Cytochrome P450
Research Area Cancer
Indications Castration-resistant Prostate Cancer

Clinical Information

Product Name Sponsor & Collaborators Indications Start Date End Date Phase
VT-464 (racemate) Viamet Pharmaceuticals, Inc. Castration-resistant Prostate Cancer 2013/12/06 Phase 2 Clinical
VT-464 (racemate) - No Development Reported

Chemical Information

M.Wt Formula CAS No. Synonyms
399.34 C18H17F4N3O3 1375603-36-3 VT464 racemate;VT 464 racemate; 1-(6,7-bis(difluoromethoxy)naphthalen-2-yl)-2-methyl-1-(1H-1,2,3-triazol-4-yl)propan-1-ol

Structure Information of VT-464 (racemate)

Smiles FC(F)OC1=C(OC(F)F)C=C(C=CC(C(C2=CNN=N2)(C(C)C)O)=C3)C3=C1
InChI InChI=1S/C18H17F4N3O3/c1-9(2)18(26,15-8-23-25-24-15)12-4-3-10-6-13(27-16(19)20)14(28-17(21)22)7-11(10)5-12/h3-9,16-17,26H,1-2H3,(H,23,24,25)

Related Products

Other Form Products of VT-464 (racemate)

Name CAS Formula Suppliers
VT-464 1610537-15-9 C18H17F4N3O3 7
VT-464 (R enantiomer) 1375603-38-5 C18H17F4N3O3 4

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Recommended Products in the Same Indication

Name CAS Formula Suppliers
VT-464 1610537-15-9 C18H17F4N3O3 7

Chemical and Physical Properties

Appearance: Melting point:
Boiling point: Flash Point:
Water Solubility: Solubility:
Density: Merck:
BRN: Refractive Index:
Vapour: EINECS:
Optical Rotation: alpha:

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