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Eltoprazine

(CAS: 98224-03-4)

Suppliers of Eltoprazine

Company Name Email Tel Country
BOC Sciences [email protected] 1-631-504-6093

Fax: 1-631-614-7828Purity: >98 % Brand: BOC Sciences

CHEMSCENE, LLC [email protected] 732-484-9848 USA

Fax: 888-484-5008Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()

MedChemexpress Co., Ltd. [email protected] 609-228-6898 USA

Fax: 609-228-5909Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()
Quality Control & MSDS Files: HNMR LCMS

Pure Chemistry Scientific Inc. [email protected] 857-928-2050 / 857-366-6788 USA

Fax: 617-206-9595Purity: 90% Brand:

Price and Availability: USD91/1g (In stock)

Shanghai Haoyuan Chemexpress Co., Ltd. [email protected] +86 (21) 5187-0955 / +86 (21) 5895-5995 China

Fax: +86 (21) 5895-5996Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()

Toronto Research Chemicals Inc. [email protected] +1 (416) 665-9696 Canada

Fax: +1 (416) 665-4439Purity: Brand:

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Background Information of Eltoprazine

Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor. IC50 value: Target: 5-HT1A/1B agonist; 5-HT2C antagonist in vitro: The binding of [3H]eltoprazine to whole tissue sections was saturable and revealed an apparent dissociation constant (Kd) of 11 nM.

Solubility of Eltoprazine

Solubility Sources
DMSO MedChemexpress Co., Ltd.

Storage Condition of Eltoprazine

Storage Condition Sources

MSDS Information

MSDS Sources

Quality Control and Spectral Data

QC Reports Sources
[HNMR] [LCMS] MedChemexpress Co., Ltd.

Mechanism and Indications

Signaling Pathways Neuronal Signaling GPCR/G Protein
Target 5-HT Receptor
Research Area Neurological Disease
Indications Cognitive Impairment Schizophrenia

Clinical Information

Product Name Sponsor & Collaborators Indications Start Date End Date Phase
Eltoprazine PsychoGenics Inc. Cognitive Impairment 2010/12/21 2012/5/01 Phase 2 Clinical
Eltoprazine PsychoGenics Inc. Schizophrenia 2010/12/21 2012/5/01 Phase 2 Clinical
Eltoprazine - Phase 2

Chemical Information

M.Wt Formula CAS No. Synonyms
220.27 C12H16N2O2 98224-03-4 DU-28853;DU28853;DU 28853; 1-(2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine

Structure Information of Eltoprazine

Smiles N1(C2=C3OCCOC3=CC=C2)CCNCC1
InChI InChI=1S/C12H16N2O2/c1-2-10(14-6-4-13-5-7-14)12-11(3-1)15-8-9-16-12/h1-3,13H,4-9H2

Related Products

Other Form Products of Eltoprazine

Name CAS Formula Suppliers
Eltoprazine (hydrochloride) 98206-09-8 C12H17ClN2O2 8

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Chemical and Physical Properties

Appearance:White to off-white Solid Melting point:
Boiling point: Flash Point:
Water Solubility: Solubility:
Density: Merck:
BRN: Refractive Index:
Vapour: EINECS:
Optical Rotation: alpha:

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