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Eltoprazine (hydrochloride)

(CAS: 98206-09-8)

Suppliers of Eltoprazine (hydrochloride)

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BOC Sciences [email protected] 1-631-504-6093

Fax: 1-631-614-7828Purity: >98 % Brand: BOC Sciences

CHEMSCENE, LLC [email protected] 732-484-9848 USA

Fax: 888-484-5008Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()

Carbosynth Limited [email protected] +44 (1635) 578-444

Fax: +44 (1635) 579-444Purity: Brand:

Price and Availability: USD132/25mg ()

Cayman Chemical Company [email protected] Toll Free (USA and Canada Only): (800) 364-9897; Direct: (734) 971-3335;Technical Support Toll Free (USA and Canada Only): (888) 526-5351;Technical Support Direct: (734) 975-3888 USA

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Price and Availability: USD25/1mg ()

MedChemexpress Co., Ltd. [email protected] 609-228-6898 USA

Fax: 609-228-5909Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()
Quality Control & MSDS Files: MSDS CoA HNMR LCMS

Shanghai Haoyuan Chemexpress Co., Ltd. [email protected] +86 (21) 5187-0955 / +86 (21) 5895-5995 China

Fax: +86 (21) 5895-5996Purity: Brand:

Price and Availability: USD110/10mg () USD422/50mg ()

Tocris Bioscience Inc. [email protected]; [email protected] +1 (636) 207-7651 USA

Fax: +1 (636) 207-7683Purity: Brand:

Price and Availability: USD125/10mg ()

Toronto Research Chemicals Inc. [email protected] +1 (416) 665-9696 Canada

Fax: +1 (416) 665-4439Purity: Brand:

Price and Availability: USD175/5mg ()

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Background Information of Eltoprazine (hydrochloride)

Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor. IC50 value: Target: 5-HT1A/1B agonist; 5-HT2C antagonist in vitro: The binding of [3H]eltoprazine to whole tissue sections was saturable and revealed an apparent dissociation constant (Kd) of 11 nM.

Solubility of Eltoprazine (hydrochloride)

Solubility Sources

Storage Condition of Eltoprazine (hydrochloride)

Storage Condition Sources

MSDS Information

MSDS Sources
MedChemexpress Co., Ltd.

Quality Control and Spectral Data

QC Reports Sources
[CoA] [HNMR] [LCMS] MedChemexpress Co., Ltd.

Mechanism and Indications

Signaling Pathways Neuronal Signaling GPCR/G Protein
Target 5-HT Receptor
Research Area Neurological Disease
Indications Cognitive Impairment Schizophrenia

Clinical Information

Product Name Sponsor & Collaborators Indications Start Date End Date Phase
Eltoprazine (hydrochloride) PsychoGenics Inc. Cognitive Impairment 2010/12/21 2012/5/01 Phase 2 Clinical
Eltoprazine (hydrochloride) PsychoGenics Inc. Schizophrenia 2010/12/21 2012/5/01 Phase 2 Clinical
Eltoprazine (hydrochloride) - No Development Reported

Chemical Information

M.Wt Formula CAS No. Synonyms
256.73 C12H17ClN2O2 98206-09-8 DU-28853 hydrochloride;DU28853 hydrochloride;DU 28853 hydrochloride; 1-(2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine hydrochloride

Structure Information of Eltoprazine (hydrochloride)

Smiles [H]Cl.N1(C2=C3OCCOC3=CC=C2)CCNCC1
InChI InChI=1S/C12H16N2O2.ClH/c1-2-10(14-6-4-13-5-7-14)12-11(3-1)15-8-9-16-12;/h1-3,13H,4-9H2;1H

Related Products

Other Form Products of Eltoprazine (hydrochloride)

Name CAS Formula Suppliers
Eltoprazine 98224-03-4 C12H16N2O2 6

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Chemical and Physical Properties

Appearance: Melting point:
Boiling point: Flash Point:
Water Solubility: Solubility:
Density: Merck:
BRN: Refractive Index:
Vapour: EINECS:
Optical Rotation: alpha:

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