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(CAS: 1532533-67-7)

Suppliers of TGR-1202

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AbMole BioScience [email protected] 1-800-660-8580 USA

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AdooQ BioScience, LLC [email protected] 855-GO-ADOOQ (855-462-3667) (US & Canada Toll Free) 866-930-6790 (US & Canada Toll Free) +1-323-389-9269 (Outside of US & Canada) USA

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Biochempartner Co., Ltd [email protected] 0086-13720134139; 0086-15971444841 China

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CHEMSCENE, LLC [email protected] 732-484-9848 USA

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MedChemexpress Co., Ltd. [email protected] 609-228-6898 USA

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Shanghai Haoyuan Chemexpress Co., Ltd. [email protected] +86 (21) 5187-0955 / +86 (21) 5895-5995 China

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Toronto Research Chemicals Inc. [email protected] +1 (416) 665-9696 Canada

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Background Information of TGR-1202

TGR-1202 is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Also active against CK1ε, with an EC50 value of 6.0 μM.

Solubility of TGR-1202

Solubility Sources
10mM in DMSO MedChemexpress Co., Ltd.

Storage Condition of TGR-1202

Storage Condition Sources
Store in a tightly closed container, in a cool and dry place. MedChemexpress Co., Ltd.

MSDS Information

MSDS Sources
MedChemexpress Co., Ltd.

Quality Control and Spectral Data

QC Reports Sources
[HNMR] [LCMS] [NP-HPLC] MedChemexpress Co., Ltd.

Mechanism and Indications

Signaling Pathways PI3K/Akt/mTOR
Target PI3K
Research Area Cancer
Indications Non-Hodgkin's Lymphoma Chronic Lymphocytic Leukemia Peripheral T-Cell Lymphoma Hodgkin's Lymphoma

Clinical Information

Product Name Sponsor & Collaborators Indications Start Date End Date Phase
TGR-1202 TG Therapeutics, Inc. Non-Hodgkin's Lymphoma Chronic Lymphocytic Leukemia Peripheral T-Cell Lymphoma Hodgkin's Lymphoma 2013/1/09 2015/10/01 Phase 1 Clinical
TGR-1202 - Phase 3

Chemical Information

M.Wt Formula CAS No. Synonyms
571.55 C31H24F3N5O3 1532533-67-7 TGR 1202;TGR1202; (S)-2-(1-(4-amino-3-(3-fluoro-4-isopropoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)ethyl)-6-fluoro-3-(3-fluorophenyl)-4H-chromen-4-one

Structure Information of TGR-1202

Smiles O=C1C(C2=CC=CC(F)=C2)=C([[email protected]@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16
InChI InChI=1S/C31H24F3N5O3/c1-15(2)41-24-9-7-18(12-22(24)34)27-26-30(35)36-14-37-31(26)39(38-27)16(3)29-25(17-5-4-6-19(32)11-17)28(40)21-13-20(33)8-10-23(21)42-29/h4-16H,1-3H3,(H2,35,36,37)/t16-/m0/s1

Related Products

Other Form Products of TGR-1202

Name CAS Formula Suppliers
TGR-1202 sulfate 1532533-75-7 C31H26F3N5O7S 2
TGR-1202 (4-methylbenzenesulfonate) 1532533-72-4 C38H32F3N5O6S 2
TGR-1202 R-enantiomer 1532533-69-9 C31H24F3N5O3 5
TGR-1202 racemate 1532533-65-5 C31H24F3N5O3 2
TGR-1202 hydrochloride 1532533-78-0 C31H25ClF3N5O3 9

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Recommended Products in the Same Indication

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TGR-1202 hydrochloride 1532533-78-0 C31H25ClF3N5O3 9

Chemical and Physical Properties

Appearance:White to off-white Solid Melting point:
Boiling point: Flash Point:
Water Solubility: Solubility:In vitro:DMSO,100 mg/mLwarmed(174.96 mM);In vitro:Ethanol,7 mg/mLwarmed(12.24 mM);In vitro:Water,Insoluble;In vivo:Add solvents to the product individually and in order(Data is from Selleck tests instead of citations):2% DMSO+30% PEG 300+2% Tween 80+H2OFo
Density: Merck:
BRN: Refractive Index:
Vapour: EINECS:
Optical Rotation: alpha:

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